{"id":24222,"date":"2021-03-18T07:29:17","date_gmt":"2021-03-18T12:29:17","guid":{"rendered":"https:\/\/blogs.funiber.org\/pt\/?p=24222"},"modified":"2021-03-18T07:29:17","modified_gmt":"2021-03-18T12:29:17","slug":"funiber-farmaco-alzheimer","status":"publish","type":"post","link":"https:\/\/www.funiber.blog\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer","title":{"rendered":"Novo f\u00e1rmaco na luta contra a doen\u00e7a de Alzheimer"},"content":{"rendered":"<p><b>Um novo f\u00e1rmaco para combater o mal de Alzheimer foi identificado por pesquisadores da Escola de Medicina da Universidade da Carolina e do Hospital Geral de Massachusetts.<\/b><\/p>\n<p><span style=\"font-weight: 400;\">O estudo foi publicado no <\/span><a href=\"https:\/\/rupress.org\/jem\" target=\"_blank\" rel=\"noopener noreferrer\"><span style=\"font-weight: 400;\">Journal of Experimental Medicine (JEM)<\/span><\/a><span style=\"font-weight: 400;\"> e afirma a efic\u00e1cia do medicamento em roedores e macacos. Se n\u00e3o forem encontrados eventos adversos, os ensaios cl\u00ednicos em humanos poder\u00e3o ser realizados em breve.\u00a0<\/span><!--more--><\/p>\n<p><b>Modulando os n\u00edveis de Abeta42<\/b><\/p>\n<p><b>Foi demonstrado que o f\u00e1rmaco modula, em vez de inibir, uma enzima chave na forma\u00e7\u00e3o de placas amiloides no c\u00e9rebro<\/b><span style=\"font-weight: 400;\">. Estas placas s\u00e3o comuns em pacientes com muta\u00e7\u00f5es que os predisp\u00f5em ao mal de Alzheimer. S\u00e3o compostos de fragmentos de prote\u00ednas, chamados de pept\u00eddeos beta-amiloides (Abeta). Entre os mais nocivos est\u00e1 o <\/span><b>Abeta42.<\/b><span style=\"font-weight: 400;\"> Por sua vez, os pept\u00eddeos s\u00e3o gerados por enzimas beta-secretase e gama-secretase.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">At\u00e9 agora, foram feitas tentativas para prevenir a doen\u00e7a, inibindo ambas as enzimas. Entretanto, ainda n\u00e3o se mostraram eficazes porque tanto a beta-secretase quanto a gama-secretase s\u00e3o indispens\u00e1veis para clivar prote\u00ednas vitais no c\u00e9rebro e outros \u00f3rg\u00e3os.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Como alternativa \u00e0 inibi\u00e7\u00e3o, foram desenvolvidos moduladores gama-secretase (GSMs) para diminuir a produ\u00e7\u00e3o de Abeta42 em at\u00e9 70%. Este mecanismo de modula\u00e7\u00e3o, em doses baixas e repetidas, demonstrou ser seguro em camundongos e macacos.<\/span><\/p>\n<p><b>O futuro do f\u00e1rmaco<\/b><\/p>\n<p><span style=\"font-weight: 400;\">Rudolph E. Tanzi, professor de neurologia em Harvard, diz que, com o estudo, \u201ctemos caracterizado farmacologicamente um potente GSM que, com base em seus atributos pr\u00e9-cl\u00ednicos, parece combinar ou exceder a efic\u00e1cia de qualquer GSM previamente testado\u201d. E, ele acrescenta esperan\u00e7osamente, se o medicamento acabar cumprindo todos os requisitos de seguran\u00e7a, <\/span><b>poderia ser usado tanto para tratar a doen\u00e7a quanto para preveni-la<\/b><span style=\"font-weight: 400;\">.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Isto se refere ao uso em pacientes com muta\u00e7\u00f5es gen\u00e9ticas que aumentam sua predisposi\u00e7\u00e3o para o mal de Alzheimer. Mas tamb\u00e9m aos casos em que as placas amiloide foram localizadas gra\u00e7as \u00e0 exames cerebrais.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Nesse sentido, a <\/span><a href=\"https:\/\/www.funiber.org.br\/\" target=\"_blank\" rel=\"noopener noreferrer\"><span style=\"font-weight: 400;\">FUNIBER<\/span><\/a><span style=\"font-weight: 400;\"> patrocina uma variedade de programas universit\u00e1rios focados em fornecer aos profissionais informa\u00e7\u00f5es abrangentes e atuais sobre os avan\u00e7os em sa\u00fade que melhoram a qualidade das pessoas idosas. Um dos cursos oferecidos \u00e9 o\u00a0<\/span><a href=\"https:\/\/www.funiber.org.br\/mestrado-em-gerontologia\" target=\"_blank\" rel=\"noopener noreferrer\"><span style=\"font-weight: 400;\">Mestrado em Gerontologia<\/span><\/a><span style=\"font-weight: 400;\">.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Fonte: <\/span><a href=\"https:\/\/www.infosalus.com\/mayores\/noticia-identifican-nuevo-farmaco-podria-prevenir-alzheimer-20210303081639.html\" target=\"_blank\" rel=\"noopener noreferrer\"><span style=\"font-weight: 400;\">Identifican un nuevo f\u00e1rmaco que podr\u00eda prevenir el Alzheimer<\/span><\/a><\/p>\n<p><span style=\"font-weight: 400;\">Foto: todos os direitos reservados.\u00a0<\/span><\/p>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Um novo f\u00e1rmaco para combater o mal de Alzheimer foi identificado por pesquisadores da Escola de Medicina da Universidade da Carolina e do Hospital Geral de Massachusetts. O estudo foi publicado no Journal of Experimental Medicine (JEM) e afirma a efic\u00e1cia do medicamento em roedores e macacos. Se n\u00e3o forem encontrados eventos adversos, os ensaios [&hellip;]<\/p>\n","protected":false},"author":10,"featured_media":24223,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"jetpack_post_was_ever_published":false,"_jetpack_newsletter_access":"","_jetpack_newsletter_tier_id":0,"footnotes":"","jetpack_publicize_message":"","jetpack_is_tweetstorm":false,"jetpack_publicize_feature_enabled":true,"jetpack_social_post_already_shared":true,"jetpack_social_options":{"image_generator_settings":{"template":"highway","enabled":false}}},"categories":[1],"tags":[108,1242,306,855,285,408,100,119,7029,248,911,267,671,2240,641,255,132,4277,113,217],"jetpack_publicize_connections":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.7 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Novo f\u00e1rmaco na luta contra a doen\u00e7a de Alzheimer<\/title>\n<meta name=\"description\" content=\"Um novo f\u00e1rmaco para combater o mal de Alzheimer foi identificado por pesquisadores da Escola de Medicina da Universidade da Carolina e do Hospital Geral de Massachusetts.\" \/>\n<meta name=\"robots\" content=\"noindex, nofollow\" \/>\n<meta property=\"og:locale\" content=\"pt_BR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Novo f\u00e1rmaco na luta contra a doen\u00e7a de Alzheimer\" \/>\n<meta property=\"og:description\" content=\"Um novo f\u00e1rmaco para combater o mal de Alzheimer foi identificado por pesquisadores da Escola de Medicina da Universidade da Carolina e do Hospital Geral de Massachusetts.\" \/>\n<meta property=\"og:url\" content=\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer\" \/>\n<meta property=\"og:site_name\" content=\"FuniBlogs - FUNIBER\" \/>\n<meta property=\"article:publisher\" content=\"https:\/\/www.facebook.com\/funiber\" \/>\n<meta property=\"article:published_time\" content=\"2021-03-18T12:29:17+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/blogs.funiber.org\/pt\/wp-content\/uploads\/2021\/03\/funiber-farmaco-alzheimer.jpg\" \/>\n\t<meta property=\"og:image:width\" content=\"570\" \/>\n\t<meta property=\"og:image:height\" content=\"350\" \/>\n\t<meta property=\"og:image:type\" content=\"image\/jpeg\" \/>\n<meta name=\"author\" content=\"Michelle\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:creator\" content=\"@FUNIBER\" \/>\n<meta name=\"twitter:site\" content=\"@FUNIBER\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"Michelle\" \/>\n\t<meta name=\"twitter:label2\" content=\"Est. tempo de leitura\" \/>\n\t<meta name=\"twitter:data2\" content=\"2 minutos\" \/>\n<script type=\"application\/ld+json\" class=\"yoast-schema-graph\">{\"@context\":\"https:\/\/schema.org\",\"@graph\":[{\"@type\":\"Article\",\"@id\":\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer#article\",\"isPartOf\":{\"@id\":\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer\"},\"author\":{\"name\":\"Michelle\",\"@id\":\"https:\/\/blogs.funiber.org\/pt\/#\/schema\/person\/a1eaaa5e57eac866a8c5946946bcf80d\"},\"headline\":\"Novo f\u00e1rmaco na luta contra a doen\u00e7a de Alzheimer\",\"datePublished\":\"2021-03-18T12:29:17+00:00\",\"dateModified\":\"2021-03-18T12:29:17+00:00\",\"mainEntityOfPage\":{\"@id\":\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer\"},\"wordCount\":412,\"publisher\":{\"@id\":\"https:\/\/blogs.funiber.org\/pt\/#organization\"},\"keywords\":[\"Alzheimer\",\"Bolsas\",\"Doen\u00e7a\",\"Doutorado\",\"Educa\u00e7\u00e3o\",\"Educa\u00e7\u00e3o a Dist\u00e2ncia\",\"Envelhecimento\",\"Estudos\",\"f\u00e1rmaco\",\"Funiber\",\"FUNIBER Opini\u00f5es\",\"Idosos\",\"mestrado\",\"Neurologia\",\"Opini\u00e3o FUNIBER\",\"Opini\u00f5es Funiber\",\"Preven\u00e7\u00e3o\",\"rem\u00e9dio\",\"Sa\u00fade\",\"Terceira idade\"],\"articleSection\":[\"Gerontologia\"],\"inLanguage\":\"pt-BR\"},{\"@type\":\"WebPage\",\"@id\":\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer\",\"url\":\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer\",\"name\":\"Novo f\u00e1rmaco na luta contra a doen\u00e7a de Alzheimer\",\"isPartOf\":{\"@id\":\"https:\/\/blogs.funiber.org\/pt\/#website\"},\"datePublished\":\"2021-03-18T12:29:17+00:00\",\"dateModified\":\"2021-03-18T12:29:17+00:00\",\"description\":\"Um novo f\u00e1rmaco para combater o mal de Alzheimer foi identificado por pesquisadores da Escola de Medicina da Universidade da Carolina e do Hospital Geral de Massachusetts.\",\"breadcrumb\":{\"@id\":\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer#breadcrumb\"},\"inLanguage\":\"pt-BR\",\"potentialAction\":[{\"@type\":\"ReadAction\",\"target\":[\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer\"]}]},{\"@type\":\"BreadcrumbList\",\"@id\":\"https:\/\/blogs.funiber.org\/pt\/gerontologia\/2021\/03\/18\/funiber-farmaco-alzheimer#breadcrumb\",\"itemListElement\":[{\"@type\":\"ListItem\",\"position\":1,\"name\":\"In\u00edcio\",\"item\":\"https:\/\/blogs.funiber.org\/pt\"},{\"@type\":\"ListItem\",\"position\":2,\"name\":\"Novo f\u00e1rmaco na luta contra a doen\u00e7a de Alzheimer\"}]},{\"@type\":\"WebSite\",\"@id\":\"https:\/\/blogs.funiber.org\/pt\/#website\",\"url\":\"https:\/\/blogs.funiber.org\/pt\/\",\"name\":\"FuniBlogs - 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